Product Name :
(R)-CE3F4
Description:
(R)-CE3F4 is a potent and selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1), with an IC50 of 4.2 μM, with 10-fold selectivity for Epac1 over Epac2 (IC50, 44 μM). (R)-CE3F4 is more potent than racemic CE3F4 and (S)-CE3F4.
CAS:
1593478-56-8
Molecular Weight:
351.01
Formula:
C11H10Br2FNO
Chemical Name:
(2R)-5,7-dibromo-6-fluoro-2-methyl-1,2,3,4-tetrahydroquinoline-1-carbaldehyde
Smiles :
C[C@@H]1CCC2=C(C=C(Br)C(F)=C2Br)N1C=O
InChiKey:
ZZLQPWXVZCPUGC-ZCFIWIBFSA-N
InChi :
InChI=1S/C11H10Br2FNO/c1-6-2-3-7-9(15(6)5-16)4-8(12)11(14)10(7)13/h4-6H,2-3H2,1H3/t6-/m1/s1
Purity:
≥98% (or refer to the Certificate of Analysis)
Shipping Condition:
Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis
Storage Condition :
Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.
Shelf Life:
≥12 months if stored properly.
Stock Solution Storage:
0 – 4 oC for 1 month or refer to the Certificate of Analysis.
Additional information:
(R)-CE3F4 is a potent and selective inhibitor of exchange protein directly activated by cAMP isoform 1 (Epac1), with an IC50 of 4.{{Diacerein} site|{Diacerein} Immunology/Inflammation|{Diacerein} Biological Activity|{Diacerein} In Vitro|{Diacerein} manufacturer|{Diacerein} Autophagy} 2 μM, with 10-fold selectivity for Epac1 over Epac2 (IC50, 44 μM).{{Picaridin} MedChemExpress|{Picaridin} Parasite|{Picaridin} Purity & Documentation|{Picaridin} In Vivo|{Picaridin} supplier|{Picaridin} Cancer} (R)-CE3F4 is more potent than racemic CE3F4 and (S)-CE3F4.|Product information|CAS Number: 1593478-56-8|Molecular Weight: 351.01|Formula: C11H10Br2FNO|Chemical Name: (2R)-5,7-dibromo-6-fluoro-2-methyl-1,2,3,4-tetrahydroquinoline-1-carbaldehyde|Smiles: C[C@@H]1CCC2=C(C=C(Br)C(F)=C2Br)N1C=O|InChiKey: ZZLQPWXVZCPUGC-ZCFIWIBFSA-N|InChi: InChI=1S/C11H10Br2FNO/c1-6-2-3-7-9(15(6)5-16)4-8(12)11(14)10(7)13/h4-6H,2-3H2,1H3/t6-/m1/s1|Technical Data|Appearance: Solid Power|Purity: ≥98% (or refer to the Certificate of Analysis)|Shipping Condition: Shipped under ambient temperature as non-hazardous chemical or refer to Certificate of Analysis|Storage Condition: Dry, dark and -20 oC for 1 year or refer to the Certificate of Analysis.PMID:25818744 |Shelf Life: ≥12 months if stored properly.|Stock Solution Storage: 0 – 4 oC for 1 month or refer to the Certificate of Analysis.|Drug Formulation: To be determined|HS Tariff Code: 382200|Products are for research use only. Not for human use.|